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4th generation nonsteroidal aromatase inhibitors: An iterative SAR-guided design, synthesis, and biological evaluation towards picomolar dual binding inhibitors |
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| Ahmed G. Eissa, Denise Barrow, Julia Gee, Lauren E. Powell, Paul A. Foster, Claire Simons |
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Design, synthesis and evaluation of novel 1,2,4-triazole derivatives as promising anticancer agents |
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| Leila Emami, Sara Sadeghian, Ayyub Mojaddami, Soghra khabnadideh, Amirhossein Sakhteman, Hossein Sadeghpour, Zeinab Faghih, Masood Fereidoonnezhad, Zahra Rezaei |
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| Ratchanok Pingaew, Vanida Choomuenwai, Ronnakorn Leechaisit, Veda Prachayasittikul, Supaluk Prachayasittikul, Virapong Prachayasittikul |
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| Pedro Alves Bezerra Morais, Carla Santana Francisco, Heberth de Paula, Rayssa Ribeiro, Mariana Alves Eloy, Clara Lirian Javarini, Álvaro Cunha Neto, Valdemar Lacerda Júnior |
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Synthesis and docking study of benzimidazole–triazolothiadiazine hybrids as aromatase inhibitors |
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| Ulviye Acar Çevik,Begüm N. Saglik,Derya Osmaniye,Serkan Levent,Betül Kaya Çavusoglu,Abdullah B. Karaduman,Yusuf Özkay,Zafer A. Kaplancikli |
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| Zeinab Faghih,Abdollah Neshat,Piero Mastrorilli,Vito Gallo,Zahra Faghih,Shirin Gilanchi |
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Design, synthesis, molecular docking, biological evaluations and QSAR studies of novel dichloroacetate analogues as anticancer agent |
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| Masood Fereidoonnezhad,S. Mohammad Hossein Tabaei,Amirhossein Sakhteman,Hassan Seradj,Zeinab Faghih,Zahra Faghih,Ayyub Mojaddami,Batool Sadeghian,Zahra Rezaei |
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Synthesis, Docking Studies and Biological Activity of New Benzimidazole- Triazolothiadiazine Derivatives as Aromatase Inhibitor |
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| Ulviye Acar Çevik,Betül Kaya Çavusoglu,Begüm Nurpelin Saglik,Derya Osmaniye,Serkan Levent,Sinem Ilgin,Yusuf Özkay,Zafer Asim Kaplancikli |
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Click chemistry in silico, docking, quantum chemical calculations, and molecular dynamics simulations to identify novel 1,2,4-triazole-based compounds as potential aromatase inhibitors |
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| Alexander M. Andrianov,Grigory I. Nikolaev,Yuri V. Kornoushenko,Sergei A. Usanov |
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Novel triazole-tetrahydroisoquinoline hybrids as human aromatase inhibitors |
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| Chanamon Chamduang,Ratchanok Pingaew,Veda Prachayasittikul,Supaluk Prachayasittikul,Somsak Ruchirawat,Virapong Prachayasittikul |
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| Sumit Kumar,Gabriella Palma,Shanen Perumal,Mandeep Kaur,Ashona Singh-Pillay,Raghu Raj,Parvesh Singh,Vipan Kumar |
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Preclinical evaluation of exemestane as a novel chemotherapy for gastric cancer |
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| Juan-Cheng Yang,Ning Chang,Deng-Chyang Wu,Wei-Chung Cheng,Wei-Min Chung,Wei-Chun Chang,Fu-Ju Lei,Chung-Jung Liu,I-Chen Wu,Hsueh-Chou Lai,Wen-Lung Ma |
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Molecular Modeling Of Novel Non-Steroidal Aromatase Inhibitors Containing 1,2,4-Triazole |
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Polyphenolic natural products and natural product-inspired steroidal mimics as aromatase inhibitors |
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| Alexander J. Nielsen,James McNulty |
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Synthesis, structural characterization, biological evaluation and molecular docking studies of new platinum(ii) complexes containing isocyanides |
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| Masood Fereidoonnezhad,Hamid R. Shahsavari,Sedigheh Abedanzadeh,Ali Nezafati,Ali Khazali,Piero Mastrorilli,Mojgan Babaghasabha,James Webb,Zeinab Faghih,Zahra Faghih,Samira Bahemmat,M. Hassan Beyzavi |
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Cycloplatinated(ii) complexes bearing an O,S-heterocyclic ligand: search for anticancer drugs |
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| Masood Fereidoonnezhad,Zahra Ramezani,Mahshid Nikravesh,Jalalaldin Zangeneh,Mohsen Golbon Haghighi,Zahra Faghih,Behrouz Notash,Hamid R. Shahsavari |
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COMPUTER-AIDED DESIGN OF POTENTIAL AROMATASE INHIBITORS BASED ON 1,2,4-TRIAZOLE DERIVATIVES |
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| A. M. Andrianov,G. I. Nikolaev,I. A. Kashyn,Yu. V. Kornoushenko,S. A. Usanov |
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